Conrad R. Burkholder

Université Claude Bernard Lyon 1 — France

Pharmacology, Toxicology and Pharmaceutics · Life Sciences

18h-index873citations55works0.02yr avg
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Research Topics

Fluorine in Organic Chemistry(47), Synthesis and Reactions of Organic Compounds(18), Synthesis and Biological Evaluation(17), Cyclopropane Reaction Mechanisms(13), Organic Chemistry Cycloaddition Reactions(12)

Publications55 total

Electron Transfer Methodologies to the Synthesis of Organo‐Fluorine Compounds
ChemInform·2005· 1 cited
ChemInform Abstract: Synthesis and Reactivity of Halogeno‐Difluoromethyl Aromatics and Heterocycles. Application to the Synthesis of gem‐Difluorinated Bioactive Compounds
ChemInform·2001
ChemInform Abstract: Synthesis of α‐(Heteroarylthio)‐α,α‐difluoroacetophenone Derivatives via the S<sub>RN</sub>1 Methodology.
ChemInform·2001
Synthesis and Electron‐Transfer Reactions of Some 3‐Difluoroacetylated Imidazo[1,2‐a]pyridine Derivatives.
ChemInform·2001
Synthesis and reactivity of halogeno-difluoromethyl aromatics and heterocycles
Journal of Fluorine Chemistry·2001· 63 cited
Synthesis of α-(heteroarylthio)-α,α-difluoroacetophenone derivatives via the SRN1 methodology
Tetrahedron Letters·2001· 18 cited
Synthesis and electron-transfer reactions of some 3-difluoroacetylated imidazo[1,2- a ]pyridine derivatives
Tetrahedron Letters·2001· 28 cited
ChemInform Abstract: The Syntheses of Nonnucleoside, HIV‐1 Reverse Transcriptase Inhibitors Containing a CF<sub>2</sub> Group. The S<sub>RN</sub>1 Reactions of 2‐(Bromodifluoromethyl)benzoxazole with the Anions Derived from Heterocyclic Thiols and Phenolic Compounds.
ChemInform·2000
The syntheses of nonnucleoside, HIV-1 reverse transcriptase inhibitors containing a CF2 group
Journal of Fluorine Chemistry·2000· 72 cited
ChemInform Abstract: Syntheses of 2‐(Bromodifluoromethyl)benzoxazole and 5‐(Bromodifluoromethyl)‐1,2,4‐oxadiazoles.
ChemInform·1999
Syntheses of 2-(bromodifluoromethyl)benzoxazole and 5-(bromodifluoromethyl)-1,2,4-oxadiazoles
Journal of Fluorine Chemistry·1999· 38 cited
ChemInform Abstract: Tetrakis(dimethylamino)ethylene (TDAE) as a Useful Reductant of Some Chlorodifluoromethylated Ketones. A New Approach for the Synthesis of α,α‐Difluoroketone Derivatives.
ChemInform·1999
ChemInform Abstract: Tetrakis(dimethylamino)ethylene as a Useful Reductant of Some Bromodifluoromethyl Heterocycles. Application to the Synthesis of New gem‐Difluorinated Heteroarylated Compounds.
ChemInform·1999
Tetrakis(dimethylamino)ethylene (TDAE) as a useful reductant of some chlorodifluoromethylated ketones. A new approach for the synthesis of α,α-difluoroketone derivatives
Tetrahedron Letters·1998· 32 cited
Tetrakis(dimethylamino)ethylene as a Useful Reductant of Some Bromodifluoromethyl Heterocycles. Application to the Synthesis of New <i>gem</i>-Difluorinated Heteroarylated Compounds
The Journal of Organic Chemistry·1998· 103 cited
ChemInform Abstract: Reaction of the 2‐(Bromodifluoromethyl)benzoxazole with Tetrakis( dimethylamino)ethylene (TDAE) in the Presence of Aldehydes. A Convenient Synthesis of 2‐(Difluoromethyl)benzoxazole Alcohols.
ChemInform·1997
Reaction of the 2-(bromodifluoromethyl)benzoxazole with tetrakis(dimethylamino)ethylene (TDAE) in the presence of aldehydes. A convenient synthesis of 2-(difluoromethyl)benzoxazole alcohols
Tetrahedron Letters·1997· 28 cited
ChemInform Abstract: The Kinetic and Thermodynamic Influence of Fluorine Versus Methyl Substituents in Methylenecyclopropane Rearrangements.
ChemInform·1996
The kinetic and thermodynamic influence of fluorine versus methyl substituents in methylenecyclopropane rearrangements
Journal of Fluorine Chemistry·1996· 12 cited
ChemInform Abstract: Synthesis of New Tetrafluorobenzo Heteroaromatic Compounds.
ChemInform·1995
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Frequent Co-authors

William R. Dolbier(45), Maurice Médebielle(14), G. E. WICKS(6), Samia Aït‐Mohand(4), Hanna Wójtowicz‐Rajchel(2), Carlos Romero(2), Khalil A. Abboud(2), David Loehle(2), Alexandre Ndedi(2), William R. Winchester(2), Gus J. Palenik(2), Marian Gawron(2), Jeffrey J. Keaffaber(2), Henryk Koroniak(2), Jyotsna Pradhan(2), George D. Purvis(2), Mark J. Seabury(2), Orland A. Soave(2), Maurice Me ́debielle(1), Rodrígo Paredes(1)