Tı́mea Imre

Centre for Social Sciences — Hungary

Chemistry · Physical Sciences

22h-index1.4kcitations73works7.02yr avg
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Research Topics

Organophosphorus compounds synthesis(20), Chemical Synthesis and Analysis(16), Click Chemistry and Applications(14), Synthesis and characterization of novel inorganic/organometallic compounds(12), Phosphorus compounds and reactions(9)

Publications73 total

Targeting a key protein-protein interaction surface on mitogen-activated protein kinases by a precision-guided warhead scaffold
Nature Communications·2024· 4 citedOpen Access
Reversible covalent c-Jun N-terminal kinase inhibitors targeting a specific cysteine by precision-guided Michael-acceptor warheads
Nature Communications·2024· 15 citedOpen Access
Site-Selective Antibody Conjugation with Dibromopyrazines
Bioconjugate Chemistry·2024· 5 citedOpen Access
Mapping protein binding sites by photoreactive fragment pharmacophores
Communications Chemistry·2024· 7 citedOpen Access
Boronic acid inhibitors of penicillin-binding protein 1b: serine and lysine labelling agents
Journal of Enzyme Inhibition and Medicinal Chemistry·2024· 4 citedOpen Access
Electrophilic MiniFrags Revealed Unprecedented Binding Sites for Covalent HDAC8 Inhibitors
Journal of Medicinal Chemistry·2023· 13 citedOpen Access
Molecular Mechanism of Labelling Functional Cysteines by Heterocyclic Thiones
ChemPhysChem·2023· 1 citedOpen Access
Mapping protein binding sites by photoreactive fragment pharmacophores
2023Open Access
Next-Generation Heterocyclic Electrophiles as Small-Molecule Covalent MurA Inhibitors
Pharmaceuticals·2022· 7 citedOpen Access
Covalent inhibitors of bacterial peptidoglycan biosynthesis enzyme MurA with chloroacetamide warhead
European Journal of Medicinal Chemistry·2022· 18 citedOpen Access
Linked PDF of Table of Contents
Synthesis·2022Open Access
A covalent strategy to target intrinsically disordered proteins: Discovery of novel tau aggregation inhibitors
European Journal of Medicinal Chemistry·2022· 19 citedOpen Access
Fragment-Sized and Bidentate (Immuno)Proteasome Inhibitors Derived from Cysteine and Threonine Targeting Warheads
Cells·2021· 8 citedOpen Access
Age-Related Inflammatory Balance Shift, Nasal Barrier Function, and Cerebro-Morphological Status in Healthy and Diseased Rodents
Frontiers in Neuroscience·2021· 7 citedOpen Access
Discovery of selective fragment-sized immunoproteasome inhibitors
European Journal of Medicinal Chemistry·2021· 14 citedOpen Access
WIDOCK: a reactive docking protocol for virtual screening of covalent inhibitors
Journal of Computer-Aided Molecular Design·2021· 29 citedOpen Access
Bromo-Cyclobutenaminones as New Covalent UDP-N-Acetylglucosamine Enolpyruvyl Transferase (MurA) Inhibitors
Pharmaceuticals·2020· 25 citedOpen Access
Assessment of Tractable Cysteines for Covalent Targeting by Screening Covalent Fragments
ChemBioChem·2020· 22 cited
An electrophilic warhead library for mapping the reactivity and accessibility of tractable cysteines in protein kinases
European Journal of Medicinal Chemistry·2020· 46 citedOpen Access
Verification of P-Glycoprotein Function at the Dermal Barrier in Diffusion Cells and Dynamic “Skin-On-A-Chip” Microfluidic Device
Pharmaceutics·2020· 34 citedOpen Access
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Frequent Co-authors

Péter Ábrányi‐Balogh(16), György M. Keserű(16), László Petri(15), Krisztina Ludányi(13), György Keglevich(13), Pál Szabó(12), Lásʐló Tőke(10), Stanislav Gobec(9), Martina Hrast(6), Krisztina Németh(5), György G. Ferenczy(5), Károly Vékey(5), H. Szelke(5), Damijan Knez(5), Aaron Keeley(5), Dávid Bajusz(4), Zoltán Márta(4), Balázs Magda(4), Melinda Sipos(4), Péter A. Szijj(3)