Akane Omagari

Kyoto University — Japan

Immunology and Microbiology · Life Sciences

9h-index911citations13works0.02yr avg
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Research Topics

HIV Research and Treatment(8), Immunotherapy and Immune Responses(4), Monoclonal and Polyclonal Antibodies Research(4), Chemokine receptors and signaling(4), vaccines and immunoinformatics approaches(4)

Publications13 total

A Point Mutation That Confers Constitutive Activity to CXCR4 Reveals That T140 Is an Inverse Agonist and That AMD3100 and ALX40-4C Are Weak Partial Agonists
Journal of Biological Chemistry·2002· 252 citedOpen Access
Certification of the Critical Importance of l-3-(2-Naphthyl)alanine at Position 3 of a Specific CXCR4 Inhibitor, T140, Leads to an Exploratory Performance of Its Downsizing Study
Bioorganic & Medicinal Chemistry·2002· 16 cited
Synthesis and evaluation of pseudopeptide analogues of a specific CXCR4 inhibitor, T140: The insertion of an (E)-alkene dipeptide isostere into the βII′-turn moiety
Bioorganic & Medicinal Chemistry Letters·2002· 30 citedOpen Access
Synthesis of Novel Anti-HIV Peptides Based on a CXCR4 Antagonist, T140, and Their SAR Study
Peptide science : proceedings of the ... Japanese Peptide Symposium·2002
Corrigendum to “conformational study of a highly specific CXCR4 inhibitor, T140, disclosing the close proximity of its intrinsic pharmacophores associated with strong anti-HIV activity”: [Bioorg. Med. Chem. Lett. 11 (2001) 359]
Bioorganic & Medicinal Chemistry Letters·2001· 12 cited
Synthesis and evaluation of bifunctional anti-HIV agents based on specific CXCR4 antagonists-AZT conjugation
Bioorganic & Medicinal Chemistry·2001· 22 cited
Development of specific CXCR4 inhibitors possessing high selectivity indexes as well as complete stability in serum based on an anti-HIV peptide T140
Bioorganic & Medicinal Chemistry Letters·2001· 109 citedOpen Access
Development of Specific CXCR4 Inhibitors Based on an Anti-HIV Peptide, T140, and Their Structure-Activity Relationships Study
Peptide science : proceedings of the ... Japanese Peptide Symposium·2001
Conformational study of a highly specific CXCR4 inhibitor, T140, disclosing the close proximity of its intrinsic pharmacophores associated with strong anti-HIV activity
Bioorganic & Medicinal Chemistry Letters·2001· 52 citedOpen Access
Pharmacophore identification of a specific CXCR4 inhibitor, T140, leads to development of effective anti-HIV agents with very high selectivity indexes
Bioorganic & Medicinal Chemistry Letters·2000· 113 citedOpen Access
Application of Ring Closing Olefin Metathesis to the Conformational Restriction of Biologically Active Peptide. Part 1
Peptide science : proceedings of the ... Japanese Peptide Symposium·2000
A Low-Molecular-Weight Inhibitor against the Chemokine Receptor CXCR4: A Strong Anti-HIV Peptide T140
Biochemical and Biophysical Research Communications·1998· 305 cited
HIV-cell Fusion Inhibitors Targeted to the HIV Second Receptor : T22 and Its Downsized Analogs with High Activity
Peptide science : proceedings of the ... Japanese Peptide Symposium·1998

Frequent Co-authors

Nobutaka Fujii(10), Hideki Nakashima(9), Akira Otaka(8), Naoki Yamamoto(8), Shinya Oishi(7), Hirokazu Tamamura(6), Hirokazu Tamamura(6), Kenichi Hiramatsu(5), Younong Xu(4), Stephen C. Peiper(4), Taisei Kanamoto(4), Toshio Hattori(3), Kazuyo Gotoh(3), Akira Otaka(3), Rieko Arakaki(2), Kenji Kanbara(2), Toshiro Ibuka(2), Nobutaka Fujii(2), Masao Matsuoka(2), Makiko Sugioka(2)