Gregory R. Bebernitz

Novartis (United States) — United States

Medicine · Health Sciences

10h-index530citations18works0.02yr avg
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Research Topics

Pancreatic function and diabetes(5), Biochemical Acid Research Studies(5), Metabolism, Diabetes, and Cancer(4), Asymmetric Synthesis and Catalysis(3), Biochemical and Molecular Research(3)

Publications18 total

Discovery of a brain-sparing GIRK1/4 inhibitor for pharmacological cardioversion of atrial fibrillation
Bioorganic & Medicinal Chemistry Letters·2023· 5 citedOpen Access
Sodium–Glucose Cotransporters
Elsevier eBooks·2016· 4 cited
P2‐059: BACE1/2 INHIBITION DOES NOT REGULATE PANCREATIC BETA CELL FUNCTION AND MASS IN MICE
Alzheimer s & Dementia·2014· 1 cited
Hepatic glycogen cycling contributes to glucose lowering effects of the glucokinase activator LCZ960
European Journal of Pharmacology·2013· 3 cited
Avoidance of the Ames test liability for aryl–amines via computation
Bioorganic & Medicinal Chemistry·2011· 32 cited
Investigation of Functionally Liver Selective Glucokinase Activators for the Treatment of Type 2 Diabetes
Journal of Medicinal Chemistry·2009· 91 cited
The Impact of Fatty Acid Oxidation on Energy Utilization: Targets and Therapy
Current Pharmaceutical Design·2002· 23 cited
Reduction in Glucose Levels in STZ Diabetic Rats by 4-(2,2-Dimethyl-1-oxopropyl)benzoic Acid:  A Prodrug Approach for Targeting the Liver.
Journal of Medicinal Chemistry·2002
The Effect of 1,3-Diaryl-[1H]-pyrazole-4-acetamides on Glucose Utilization in ob/ob Mice
Journal of Medicinal Chemistry·2001· 140 cited
Reduction in Glucose Levels in STZ Diabetic Rats by 4-(2,2-Dimethyl-1-oxopropyl)benzoic Acid:  A Prodrug Approach for Targeting the Liver
Journal of Medicinal Chemistry·2000· 13 cited
ChemInform Abstract: Anilides of (R)‐Trifluoro‐2‐hydroxy‐2‐methylpropionic Acid as Inhibitors of Pyruvate Dehydrogenase Kinase.
ChemInform·2000
Anilides of (<i>R</i>)-Trifluoro-2-hydroxy-2-methylpropionic Acid as Inhibitors of Pyruvate Dehydrogenase Kinase
Journal of Medicinal Chemistry·2000· 60 citedOpen Access
(<i>R</i>)-3,3,3-Trifluoro-2-hydroxy-2-methylpropionamides Are Orally Active Inhibitors of Pyruvate Dehydrogenase Kinase
Journal of Medicinal Chemistry·1999· 43 citedOpen Access
Hypoglycemic Prodrugs of 4-(2,2-Dimethyl-1-oxopropyl)benzoic Acid
Journal of Medicinal Chemistry·1998· 11 cited
ChemInform Abstract: A VERSATILE 3‐ACYLTETRAMIC ACID REAGENT
Chemischer Informationsdienst·1985
ChemInform Abstract: TOTAL SYNTHESIS OF (‐)‐TIRANDAMYCIN A
Chemischer Informationsdienst·1985
A versatile 3-acyltetramic acid reagent
The Journal of Organic Chemistry·1985· 21 cited
Total synthesis of (-)-tirandamycin A
Journal of the American Chemical Society·1985· 83 cited

Frequent Co-authors

Robert J. Strohschein(6), Jiaping Gao(5), Herbert F. Schuster(4), R. H. Schlessinger(4), Wieslawa Maniara(3), Thomas D. Aicher(3), Douglas C. Knorr(3), Leonard Brand(3), Jeremy G. Dain(3), Rhonda Oetting Deems(3), Alokesh Duttaroy(2), Melissa S. Grondine(2), Louise Kirman(2), Peter Lin(2), A. J. POSS(2), Suraj S. Shetty(2), Christine C. Vinluan(2), Emma L. Kaplan(2), Carol J. Dragland(2), Dominick DelGrande(2)