Stephen L. Buchwald

Massachusetts Institute of Technology — United States

Chemistry · Physical Sciences

177h-index107.0kcitations1.3kworks9.12yr avg

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Research Topics

Catalytic C–H Functionalization Methods(610), Catalytic Cross-Coupling Reactions(596), Asymmetric Hydrogenation and Catalysis(359), Asymmetric Synthesis and Catalysis(156), Chemical Synthesis and Analysis(146)

Publications1.3k total

Ligand Design Enables Cu-Catalyzed Etherification of Aryl Bromides Using Mild Bases

Organic Letters·2026Open Access

Development of a Ligand for Cu-Catalyzed Amination of Base-Sensitive (Hetero)aryl Chlorides

4 cited

Journal of the American Chemical Society·2025· 4 citedOpen Access

Copper Hydride-Catalyzed Net Hydroformylation of Unactivated Terminal Olefins

Organic Letters·2025

Developing Pharmaceutically Relevant Pd-Catalyzed C–N Coupling Reactivity Models Leveraging High-Throughput Experimentation

9 cited

Journal of the American Chemical Society·2025· 9 cited

Automated Flow Synthesis of Artificial Heme Enzymes for Enantiodivergent Biocatalysis

4 cited

Journal of the American Chemical Society·2025· 4 cited

Kinetic Modeling Enables Understanding of Off-Cycle Processes in Pd-Catalyzed Amination of Five-Membered Heteroaryl Halides

6 cited

Journal of the American Chemical Society·2024· 6 citedOpen Access

Deciphering the alteration of MAP2 interactome caused by a schizophrenia-associated phosphorylation

1 cited

Neurobiology of Disease·2024· 1 citedOpen Access

Correction to “Copper-Catalyzed Amination of Aryl Chlorides under Mild Reaction Conditions”

Journal of the American Chemical Society·2024

Identification of reactivity hotspots at the interfaces of protein–protein interactions

2024Open Access

Development of a Deactivation-Resistant Dialkylbiarylphosphine Ligand for Pd-Catalyzed Arylation of Secondary Amines

24 cited

Journal of the American Chemical Society·2024· 24 citedOpen Access

Copper-Catalyzed Amination of Aryl Chlorides under Mild Reaction Conditions

26 cited

Journal of the American Chemical Society·2024· 26 citedOpen Access

Site-Specific Antibody Prodrugs via <i>S</i> -Arylation: a Bioconjugation Approach Toward Masked Tyrosine Analogues

8 cited

Journal of the American Chemical Society·2024· 8 cited

Cu-Catalyzed Amination of Base-Sensitive Aryl Bromides and the Chemoselective N- and O-Arylation of Amino Alcohols

42 cited

Journal of the American Chemical Society·2024· 42 citedOpen Access

Automated Flow Synthesis of Artificial Heme Enzymes for Enantioselective Biocatalysis

2 cited

2024· 2 citedOpen Access

CuH-Catalyzed Regio- and Enantioselective Formal Hydroformylation of Vinyl Arenes

11 cited

Journal of the American Chemical Society·2024· 11 citedOpen Access

Miquel Pericàs – an Outstanding Scientist and a Great Friend

Advanced Synthesis & Catalysis·2024Open Access

Room‐Temperature Copper‐Catalyzed Etherification of Aryl Bromides

Angewandte Chemie·2024

Room‐Temperature Copper‐Catalyzed Etherification of Aryl Bromides

34 cited

Angewandte Chemie International Edition·2024· 34 citedOpen Access

Room-Temperature Cu-Catalyzed Etherification of Aryl Bromides

1 cited

2024· 1 citedOpen Access

Site-Specific Antibody Prodrugs via S-Arylation: A Bioconjugation Approach Toward Masked Tyrosine Analogues

1 cited

2023· 1 citedOpen Access

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Frequent Co-authors

John P. Wolfe(8), Artis Klapars(6), Xiaohua Huang(5), Jingjun Yin(4), Timothy E. Barder(3), Jon C. Antilla(3), D. Surry(2), Seble Wagaw(2), Shawn D. Walker(2), Joseph R. Martinelli(2), Bryant H. Yang(2), Anil S. Guram(2), David W. Old(2), Donald A. Watson(2), Kevin W. Anderson(2), Joseph P. Sadighi(2), Michael T. Pirnot(2), Fuk Yee Kwong(2), Paula Ruiz‐Castillo(1), Rubén Martı́n(1)