Fredrik Björkling

University of Copenhagen — Denmark

Biochemistry, Genetics and Molecular Biology · Life Sciences

32h-index4.4kcitations120works2.72yr avg
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Research Topics

Enzyme Catalysis and Immobilization(15), Chemical Synthesis and Analysis(11), Estrogen and related hormone effects(9), Analytical Chemistry and Chromatography(9), Microbial Metabolic Engineering and Bioproduction(9)

Publications119 total

SAT-317 Design and Evaluation of novel CYP17A1 Inhibitors: Potential Therapeutic Agents for Castration-Resistant Prostate Cancer
Journal of the Endocrine Society·2025Open Access
Structure-activity study of oncocins modified with cationic polar moieties at the termini
European Journal of Medicinal Chemistry Reports·2025Open Access
Steroidogenesis and CYP17A1 inhibition: development of potent inhibitors for adrenal and gonadal steroid biosynthesis
Endocrine Abstracts·2025
Design and Evaluation of Novel CYP17A1 Inhibitors: Potential Therapeutic Agents for Castration-Resistant Prostate Cancer (Abstract ID: 190110)
Journal of Pharmacology and Experimental Therapeutics·2025
Pyridine indole hybrids as novel potent CYP17A1 inhibitors
Journal of Enzyme Inhibition and Medicinal Chemistry·2025· 8 citedOpen Access
Polymyxins with Potent Antibacterial Activity against Colistin-Resistant Pathogens: Fine-Tuning Hydrophobicity with Unnatural Amino Acids
Journal of Medicinal Chemistry·2024· 8 citedOpen Access
Studies of antibacterial activity (in vitro and in vivo) and mode of action for des-acyl tridecaptins (DATs)
European Journal of Medicinal Chemistry·2023· 1 cited
Structure-activity study of oncocin: On-resin guanidinylation and incorporation of homoarginine, 4-hydroxyproline or 4,4-difluoroproline residues
Bioorganic Chemistry·2023· 10 citedOpen Access
Exploring the Potential of Sulfur Moieties in Compounds Inhibiting Steroidogenesis
Biomolecules·2023· 8 citedOpen Access
Non-steroidal CYP17A1 Inhibitors: Discovery and Assessment
Journal of Medicinal Chemistry·2023· 59 citedOpen Access
Antimicrobial Peptides Incorporating Halogenated Marine-Derived Amino Acid Substituents
ACS Medicinal Chemistry Letters·2023· 8 citedOpen Access
Selected strategies to fight pathogenic bacteria
Journal of Enzyme Inhibition and Medicinal Chemistry·2023· 48 citedOpen Access
Studies of Antibacterial Activity (in Vitro and in Vivo) and Mode of Action for Des-Acyl Tridecaptins (Dats)
SSRN Electronic Journal·2023Open Access
Synthesis and Structure–Activity Relationships of Novel Non-Steroidal CYP17A1 Inhibitors as Potential Prostate Cancer Agents
Biomolecules·2022· 22 citedOpen Access
Imitation of β-lactam binding enables broad-spectrum metallo-β-lactamase inhibitors
Nature Chemistry·2021· 77 citedOpen Access
Evaluation of 1<i>H</i>-Triazole-1-[<i>N</i>,<i>N</i>′-Bis(<i>tert</i>-butoxycarbonyl)]carboxamidine in Solution-Phase and On-Resin Guanidinylation
The Journal of Organic Chemistry·2021· 4 cited
Correction to “Structural Basis of Metallo-β-lactamase Inhibition by <i>N</i>-Sulfamoylpyrrole-2-carboxylates”
ACS Infectious Diseases·2021· 1 citedOpen Access
Peptide/β-Peptoid Hybrids with Ultrashort PEG-Like Moieties: Effects on Hydrophobicity, Antibacterial Activity and Hemolytic Properties
International Journal of Molecular Sciences·2021· 9 citedOpen Access
Structural Basis of Metallo-β-lactamase Inhibition by<i>N</i>-Sulfamoylpyrrole-2-carboxylates
ACS Infectious Diseases·2021· 28 citedOpen Access
Optimized Synthesis of Fmoc/Boc‐Protected PNA Monomers and their Assembly into PNA Oligomers.
European Journal of Organic Chemistry·2021· 14 cited
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Frequent Co-authors

Maxwell Sehested(9), Peter Buhl Jensen(8), Morten Dahl Sørensen(7), Torbjörn Norin(6), Kamille Dumong Erichsen(6), Sven Erik Godtfredsen(5), Ole Kirk(5), Karl Hult(5), Lise Binderup(5), Henrik Franzyk(5), Søren Jensby Nielsen(4), Mette Krogh Christensen(4), Mette Munk Jensen(4), Jacob Madsen(4), Liselotte Højgaard(4), Andreas Kjær(4), Uffe H. Olesen(3), John Boutelje(3), Sten Gatenbeck(3), Scilla Latini(3)