Prakash C. Taunk

Bristol-Myers Squibb (United States) — United States

Medicine · Health Sciences

8h-index1.3kcitations21works0.02yr avg
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Research Topics

Peptidase Inhibition and Analysis(7), Phenothiazines and Benzothiazines Synthesis and Activities(7), Diabetes Treatment and Management(4), Neuropeptides and Animal Physiology(4), Synthesis and Biological Evaluation(4)

Publications21 total

Potent and selective biphenyl azole inhibitors of adipocyte fatty acid binding protein (aFABP)
Bioorganic & Medicinal Chemistry Letters·2006· 150 citedOpen Access
Seco-prolinenitrile inhibitors of dipeptidyl peptidase IV define minimal pharmacophore requirements at P1
Bioorganic & Medicinal Chemistry Letters·2005· 3 citedOpen Access
Diprolyl nitriles as potent dipeptidyl peptidase IV inhibitors
Bioorganic & Medicinal Chemistry Letters·2005· 23 citedOpen Access
Discovery and Preclinical Profile of Saxagliptin (BMS-477118):  A Highly Potent, Long-Acting, Orally Active Dipeptidyl Peptidase IV Inhibitor for the Treatment of Type 2 Diabetes
Journal of Medicinal Chemistry·2005· 617 citedOpen Access
CCDC 253955: Experimental Crystal Structure Determination
The Cambridge Structural Database·2005Open Access
Synthesis of Novel Potent Dipeptidyl Peptidase IV Inhibitors with Enhanced Chemical Stability:  Interplay between the N-Terminal Amino Acid Alkyl Side Chain and the Cyclopropyl Group of α-Aminoacyl-<scp>l</scp>-<i>cis</i>-4,5-methanoprolinenitrile-Based Inhibitors
Journal of Medicinal Chemistry·2004· 103 citedOpen Access
Application of robotics to steady state enzyme kinetics: analysis of tight-binding inhibitors of dipeptidyl peptidase IV
Analytical Biochemistry·2003· 7 cited
Microsomal triglyceride transfer protein inhibitors: discovery and synthesis of alkyl phosphonates as potent MTP inhibitors and cholesterol lowering agents
Bioorganic & Medicinal Chemistry Letters·2003· 18 citedOpen Access
A Novel Series of Highly Potent Benzimidazole-Based Microsomal Triglyceride Transfer Protein Inhibitors
Journal of Medicinal Chemistry·2001· 61 citedOpen Access
An MTP Inhibitor That Normalizes Atherogenic Lipoprotein Levels in WHHL Rabbits
Science·1998· 268 cited
ChemInform Abstract: Dual Metalloprotease Inhibitors. Part 5. Utilization of Bicyclic Azepinonethiazolidines and Azepinonetetrahydrothiazines in Constrained Peptidomimetics of Mercaptoacyl Dipeptides.
ChemInform·1995
Dual metalloprotease inhibitors.v. Utilization of bicyclic azepinonethiazolidines and azepinonetetrahydrothiazines in constrained peptidomimetics of mercaptoacyl dipeptides
Bioorganic & Medicinal Chemistry Letters·1995· 30 cited
ChemInform Abstract: Synthesis of a New Benzo[a]phenothiazine Amino Alcohol as a Proposed Antimalarial.
Chemischer Informationsdienst·1986
Synthesis of a new benzo[<i>a</i>]phenothiazine amino alcohol as a proposed antimalarial
Journal of Heterocyclic Chemistry·1985· 1 cited
ChemInform Abstract: NEW TETRACYCLIC RING SYSTEMS. SYNTHESIS OF 1H‐OXAZOLO(5,4,3‐KL)PHENOTHIAZINES AND (1,4)OXAZINO(2,3,4‐KL)PHENOTHIAZINES
Chemischer Informationsdienst·1983
New tetracyclic ring systems. Synthesis of 1<i>H</i>‐oxazolo[5,4,3‐<i>kl</i>]phenothiazines and [1,4]oxazino[2,3,4‐<i>kl</i>]phenothiazines
Journal of Heterocyclic Chemistry·1982· 5 cited
ChemInform Abstract: SYNTHESES OF SOME HYDROXYLATED METABOLITES OF PSYCHOTROPIC TRIFLUOROMETHYL ANALOGS OF CHLORPROMAZINE
Chemischer Informationsdienst·1982
Syntheses of some hydroxylated metabolites of psychotropic trifluoromethyl analogs of chlorpromazine
Journal of Heterocyclic Chemistry·1981· 7 cited
ChemInform Abstract: SYNTH. VON 2‐AMINO‐5‐FLUOR‐THIOPHENOL UND SEINE UMWANDLUNG IN PHENOTHIAZINE UND DEREN SULFONE
Chemischer Informationsdienst Organische Chemie·1971
Die Synthese von 2-Amino-5-fluorthiophenol und seine Umwandlung in Phenothiazine und deren Sulfone
Monatshefte für Chemie - Chemical Monthly·1971· 8 cited
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Frequent Co-authors

Jeffrey A. Robl(10), David R. Magnin(10), Ligaya M. Simpkins(7), James G. Robertson(6), Aiying Wang(5), Lawrence G. Hamann(5), Richard Sulsky(5), R. L. Mital(5), Michael Cap(4), Scott A. Biller(4), Rex A. Parker(4), Thomas Harrity(4), Edward A. Nodiff(4), David J. Augeri(3), David A. Betebenner(3), Song‐Ping Han(3), Benoni E. Abboa‐Offei(3), Jovita Marcinkeviciene(3), Mark Kirby(3), John R. Wetterau(3)