Federico Da Settimo

University of Pisa — Italy

Chemistry · Physical Sciences

44h-index6.3kcitations364works6.32yr avg
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Research Topics

Synthesis and Characterization of Heterocyclic Compounds(56), Adenosine and Purinergic Signaling(47), Synthesis and biological activity(46), Synthesis and Biological Evaluation(41), Neuroscience and Neuropharmacology Research(39)

Publications364 total

Repurposing Auranofin for Oncology and Beyond: A Brief Overview of Clinical Trials as Mono- and Combination Therapy
Pharmaceuticals·2025Open Access
Repurposing Auranofin for Oncology and Beyond: A Brief Overview of Clinical Trials as Mono- and Combination Therapy
Preprints.org·2025Open Access
2-(Phenylamino)-7,8-dihydroquinazolin-5(6H)-one, a promising scaffold for MAO-B inhibitors with potential GSK3β targeting
European Journal of Medicinal Chemistry·2025· 1 citedOpen Access
18 kDa TSPO targeting drives polarized human microglia towards a protective and restorative neurosteroidome profile
Cellular and Molecular Life Sciences·2025· 5 citedOpen Access
Discovery of the First-in-Class Dual TSPO/Carbonic Anhydrase Modulators with Promising Neurotrophic Activity
ACS Chemical Neuroscience·2024
Discovery of <i>N</i>-substituted-2-oxoindolin benzoylhydrazines as c-MET/SMO modulators in EGFRi-resistant non-small cell lung cancer
RSC Medicinal Chemistry·2024Open Access
Pursuing Polypharmacology: Benzothiopyranoindoles as G-Quadruplex Stabilizers and Topoisomerase I Inhibitors for Effective Anticancer Strategies
ACS Medicinal Chemistry Letters·2024· 1 citedOpen Access
Enhancing the Anticancer Activity of Attenuated <i>Listeria monocytogenes</i> by Cell Wall Functionalization with “Clickable” Doxorubicin
ACS Chemical Biology·2024· 10 citedOpen Access
TSPO Radioligands for Neuroinflammation: An Overview
Molecules·2024· 21 citedOpen Access
Indole-Based Compounds in the Development of Anti-Neurodegenerative Agents
Molecules·2024· 38 citedOpen Access
Human oligodendrocyte-like cell differentiation is promoted by TSPO-mediated endogenous steroidogenesis
Biochimica et Biophysica Acta (BBA) - Molecular Basis of Disease·2024· 5 citedOpen Access
Enhancing the Anticancer Activity of Attenuated Listeria monocytogenes by Cell Wall Functionalization with 'Clickable' Doxorubicin
SSRN Electronic Journal·2024Open Access
Anti‐inflammatory and anti‐apoptotic activity of a <scp>TSPO</scp> ligand in slowing retina neurodegeneration in a model of retinitis pigmentosa
Acta Ophthalmologica·2024
Targeting the Translocator Protein (18 kDa) in Cardiac Diseases: State of the Art and Future Opportunities
Journal of Medicinal Chemistry·2023· 9 citedOpen Access
Anti-Proliferative Properties of the Novel Hybrid Drug Met-ITC, Composed of the Native Drug Metformin with the Addition of an Isothiocyanate H2S Donor Moiety, in Different Cancer Cell Lines
International Journal of Molecular Sciences·2023· 12 citedOpen Access
Tyrosine kinase inhibitors (TKIs) for ovarian cancer treatment: from organic to inorganic chemotherapeutics towards selectivity—a perspective overview
BioMetals·2023· 2 citedOpen Access
Enhancing the anticancer activity of attenuated Listeria monocytogenes by cell wall functionalization with “clickable” doxorubicin
2023Open Access
Enhancing the anticancer activity of attenuated Listeria monocytogenes by cell wall functionalization with “clickable” doxorubicin
2023Open Access
A NOVEL DERIVATIVE OF 2-PHENYL-PYRIDO[1,2-a]PYRIMIDIN-4-ONE INHIBITS ENDOTHELIAL CELL DYSFUNCTION AND SMOOTH MUSCLE CELL PROLIFERATION/ACTIVATION
Zenodo (CERN European Organization for Nuclear Research)·2023Open Access
Indol-3-ylglyoxylamide as Privileged Scaffold in Medicinal Chemistry
Pharmaceuticals·2023· 4 citedOpen Access
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Frequent Co-authors

Sabrina Taliani(31), Concettina La Motta(28), Ettore Novellino(22), Claudia Martini(20), Francesca Simorini(15), Anna María Marini(15), Silvia Salerno(12), Stefania Sartini(12), Giampaolo Primofiore(12), Giovanni Greco(11), Barbara Costa(10), Elisabetta Barresi(9), Eleonora Da Pozzo(9), Antonio Lavecchia(8), Luciana Marinelli(8), Sandro Cosconati(7), A. DA SETTIMO(7), Laura Mugnaini(6), Barbara Cosimelli(6), Maria Letizia Trincavelli(6)