Nesrin Gökhan-Kelekçi

Hacettepe University — Turkey

Chemistry · Physical Sciences

9h-index897citations14works0.52yr avg
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Research Topics

Synthesis and biological activity(9), Synthesis and Biological Evaluation(6), Click Chemistry and Applications(4), Synthesis and Characterization of Heterocyclic Compounds(3), Computational Drug Discovery Methods(2)

Publications14 total

Synthesis and biological evaluation of novel naproxen–phenacetin triazole hybrids as promising anti-inflammatory agents with enhanced gastrointestinal tolerability
Bioorganic Chemistry·2025
Some novel 5-benzylidenethiazolo[3,2-b]-1,2,4-triazole-6(5H)-one derivatives in the battle against cancer: Design, synthesis and their biological activities
Journal of Molecular Structure·2024· 1 cited
Synthesis, characterization, and in vivo pharmacological evaluation of novel mannich bases derived from 1,2,4-triazole containing a naproxen moiety
Bioorganic Chemistry·2020· 26 cited
Determination of p<i>K</i><sub>a</sub> Values of Some Benzoxazoline Derivatives and the Structure–Activity Relationship
Journal of Chemical & Engineering Data·2013· 10 cited
Evaluation of selective human MAO inhibitory activities of some novel pyrazoline derivatives
Journal of Neural Transmission·2013· 15 cited
Synthesis, molecular modeling, and in vitro screening of monoamine oxidase inhibitory activities of some novel hydrazone derivatives
Journal of Neural Transmission·2013· 19 cited
Insights into the binding mode of new N-substituted pyrazoline derivatives to MAO-A: docking and quantum chemical calculations
Journal of Neural Transmission·2012· 8 cited
Synthesis, crystal structures and DFT studies of 1-[2-(5-methyl-2-benzoxazolinone-3-yl)acetyl]-3-phenyl-5-(3,4-dimethoxyphenyl)-4,5-dihydro-1H-pyrazole and 1-[2-(5-chloro-2-benzoxazolinone-3-yl)acetyl]-3-phenyl-5-(4-methoxyphenyl)-4,5-dihydro-1H-pyrazole
Journal of Molecular Structure·2011· 15 cited
Synthesis and molecular modeling of some novel hexahydroindazole derivatives as potent monoamine oxidase inhibitors
Bioorganic & Medicinal Chemistry·2009· 38 citedOpen Access
New pyrazoline bearing 4(3H)-quinazolinone inhibitors of monoamine oxidase: Synthesis, biological evaluation, and structural determinants of MAO-A and MAO-B selectivity
Bioorganic & Medicinal Chemistry·2008· 157 citedOpen Access
Molecular structure of 2-methylamino-5-[(5-methyl-2-benzoxazolinone-3-yl)methyl]-1,3,4-thiadiazole dihydrophosphate: a combined X-ray crystallographic and ab initio study
Structural Chemistry·2008· 4 cited
Synthesis and characterization of some new 2(<i>3H</i>)-benzoxazolones with analgesic and antiinflammatory activities
Journal of Enzyme Inhibition and Medicinal Chemistry·2008· 9 cited
A new therapeutic approach in Alzheimer disease: Some novel pyrazole derivatives as dual MAO-B inhibitors and antiinflammatory analgesics
Bioorganic & Medicinal Chemistry·2007· 227 citedOpen Access
1-Acylthiosemicarbazides, 1,2,4-triazole-5(4H)-thiones, 1,3,4-thiadiazoles and hydrazones containing 5-methyl-2-benzoxazolinones: Synthesis, analgesic-anti-inflammatory and antimicrobial activities
Bioorganic & Medicinal Chemistry·2007· 368 cited

Frequent Co-authors

U. Salgin-Goksen(5), Gülberk Uçar(5), Kemal Yelekçi(5), Ş. Işık(3), Ahmet Avci(3), Birsen Tozkoparan(3), Göknur Aktay(2), Samiye Yabanoğlu(2), O. Ozgen(2), Engin Kendi(2), Akgül Yeşilada(2), A. Altan Bilgin(2), Ayşe Ercan(2), Zarife Sibel Şahin(2), Hayrünnisa Taşci(2), Samiye Yabanoğlu‐Çiftçi(2), Hakkı Erdoğan(2), O. Goktas(1), Yavuz Köysal(1), Ekrem Kılıç(1)