Hideaki Kakeya

Kyoto University — Japan

Medicine · Health Sciences

49h-index9.4kcitations345works1.82yr avg
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Research Topics

Microbial Natural Products and Biosynthesis(106), Synthetic Organic Chemistry Methods(62), Chemical Synthesis and Analysis(42), Marine Sponges and Natural Products(34), Peptidase Inhibition and Analysis(20)

Publications345 total

Inhibitory Effects of Imidazole Dipeptides and 2-Oxo-Imidazole Dipeptides on Intracellular ROS Generation and Degradation of Protein and DNA
MDPI (MDPI AG)·2026Open Access
Structure Revision, Absolute Configuration Determination, and Biological Evaluation of Furanonaphthoquinone I
Journal of Natural Products·2026
Quantitative analysis of D/L-serine and D/L-proline in serum by isotope-coded derivatization using an original chiral resolution labeling reagent
Journal of Pharmaceutical and Biomedical Analysis Open·2025Open Access
Recent Advances in Bioactive Natural Products from Plant Fruits: Structures, Activities, and Future Prospects
Plant Foods for Human Nutrition·2025· 1 cited
Abstract C009: Development of an innovative anticancer drug TBP1901, an injectable prodrug of curcumin, for the treatment of multiple myeloma
Molecular Cancer Therapeutics·2025
Abstract B038: Discovery of an anticancer seed targeting cancer stem cells and analysis of its mode of action
Molecular Cancer Therapeutics·2025
Natural product-inspired chemical biology: development of highly sensitive labeling reagents for amino acids and scarce natural products
Phytochemistry Letters·2025Open Access
Recent Progress in Nonanolides of Natural Origin: Structures, Synthesis, Biosynthesis, and Bioactivities
The Chemical Record·2025· 1 cited
Identification of a key amino acid residue in the cofactor-independent oxidase ActVA-ORF3 involved in actinorhodin biosynthesis using AlphaFold2-predicted modeling and mutational analysis
Results in Chemistry·2025Open Access
Natural Lysine-Reactive Meroterpenoids, Stachybenzals A–C, as Covalent Asparagine Synthetase Inhibitors
Journal of Natural Products·2025· 3 cited
Isolation and structure determination of streptospherins B–F, novel cancer stem cell inhibitors, produced by Streptomyces sp. KUSC-240
The Journal of Antibiotics·2025· 1 cited
Formation of giant ER sheets by pentadecanoic acid causes lipotoxicity in fission yeast
Proceedings of the National Academy of Sciences·2025· 1 citedOpen Access
Winners of the 2024 Tu Youyou Award
Molecules·2025Open Access
Streptospherin A, a New Cancer Stem Cell Inhibitor, Produced by <i>Streptomyces</i> sp. KUSC-240
Chemical and Pharmaceutical Bulletin·2025· 1 citedOpen Access
A new pyranonaphthoquinone, actinoquinonal A, and its congeners from the combined-culture of Streptomyces sp. 23–50 and Tsukamurella pulmonis TP-B0596
The Journal of Antibiotics·2025· 2 cited
Discovery, total synthesis, and biological evaluation of tyrcinnamins as antibacterial agents and tyrosinase activators
European Journal of Medicinal Chemistry·2025· 4 cited
Inhibition of Surfactin Biosynthesis in <i>Bacillus Subtilis</i> Using Cell‐Permeable Adenylation Domain Inhibitors
ChemBioChem·2025Open Access
Structural Elucidation using Highly Sensitive Labeling Reagents and Total Synthesis of Amoxetamide A, a New Anoikis Inducer
Chemistry - A European Journal·2025· 2 citedOpen Access
Recent progress in chemistry and bioactivity of novel enzyme inhibitors from natural products: A comprehensive review
European Journal of Medicinal Chemistry·2025· 3 cited
Twisted Amide‐Mediated Synthesis and Rapid Structure‐Activity Relationship Study of Medium‐Sized Cyclic Peptides
Chemistry - A European Journal·2025· 1 citedOpen Access
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Frequent Co-authors

Hiroyuki Osada(28), Rie Onose(10), Mitsuru Shoji(9), Yujiro Hayashi(9), Junichiro Yamaguchi(7), Cheng‐Bin Cui(6), Yoichi Sunagawa(6), Hiromichi Wada(6), Yasufumi Katanasaka(6), Koji Hasegawa(6), Tatsuya Morimoto(6), Shinichi Nishimura(5), Atsushi Imaizumi(5), Gen Okada(4), Hiroyuki Koshino(3), Yukihiro Asami(3), Arika Yoshida(3), Masafumi Funamoto(3), Yusuke Miyazaki(3), Ryosuke Sugiyama(3)