Ravi S. Garigipati

Pfizer (United States) — United States

Biochemistry, Genetics and Molecular Biology · Life Sciences

22h-index1.6kcitations45works0.02yr avg
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Research Topics

Chemical Synthesis and Analysis(9), Synthetic Organic Chemistry Methods(9), Asymmetric Synthesis and Catalysis(8), Synthesis and biological activity(5), Microbial Natural Products and Biosynthesis(4)

Publications45 total

Identification of a novel, non-tetrahydroquinoline variant of the cholesteryl ester transfer protein (CETP) inhibitor torcetrapib, with improved aqueous solubility
Xenobiotica·2013· 4 cited
Process Development and Scale-Up of an Hsp90 Inhibitor
Organic Process Research & Development·2012· 24 cited
1P-0195 Discovery of CP-760,144: A potent synthetic antagonist of monocyte chemoattractant protein-1 (MCP-1)
Atherosclerosis Supplements·2003
Pyrimidinylimidazole inhibitors of p38: cyclic N-1 imidazole substituents enhance p38 kinase inhibition and oral activity
Bioorganic & Medicinal Chemistry Letters·2001· 105 citedOpen Access
Novel solid-phase preparation of 2,6,9-trisubstituted purines for combinatorial library generation
Tetrahedron Letters·2001· 30 cited
Reagents for combinatorial organic synthesis: preparation and uses of Rink-chloride
Tetrahedron Letters·1997· 40 cited
Enantioselective Synthesis of 5-LO Inhibitor Hydroxyureas. Tandem Nucleophilic Addition−Intramolecular Cyclization of Chiral Nitrones
The Journal of Organic Chemistry·1997· 34 cited
Novel frameworks for trifluoromethyl ketone and phosphonate tsa inhibitors of type II PLA2
Bioorganic & Medicinal Chemistry Letters·1997· 4 cited
ChemInform Abstract: Bicyclic N‐Hydroxyurea Inhibitors of 5‐Lipoxygenase: Pharmacodynamic, Pharmacokinetic, and in vitro Metabolic Studies Characterizing N‐ Hydroxy‐N‐(2,3‐dihydro‐6‐(phenylmethoxy)‐3‐benzofuranyl)urea.
ChemInform·1997
ChemInform Abstract: 1‐Substituted 4‐Aryl‐5‐pyridinylimidazoles: A New Class of Cytokine Suppressive Drugs with Low 5‐Lipoxygenase and Cyclooxygenase Inhibitory Potency.
ChemInform·1997· 6 cited
Regulation of stress-induced cytokine production by pyridinylimidazoles; inhibition of CSBP kinase
Bioorganic & Medicinal Chemistry·1997· 218 cited
An NMR Method To Identify Nondestructively Chemical Compounds Bound to a Single Solid-Phase-Synthesis Bead for Combinatorial Chemistry Applications
Journal of the American Chemical Society·1996· 120 cited
1,2-Thiazines and their Benzo Derivatives
Elsevier eBooks·1996· 7 cited
Use of Spin Echo Magic Angle Spinning <sup>1</sup>H NMR in Reaction Monitoring in Combinatorial Organic Synthesis
The Journal of Organic Chemistry·1996· 4 cited
Bicyclic N-Hydroxyurea Inhibitors of 5-Lipoxygenase:  Pharmacodynamic, Pharmacokinetic, and <i>in Vitro</i> Metabolic Studies Characterizing <i>N</i>-Hydroxy-<i>N</i>-(2,3-dihydro-6-(phenylmethoxy)-3-benzofuranyl)urea
Journal of Medicinal Chemistry·1996· 29 citedOpen Access
1-Substituted 4-Aryl-5-pyridinylimidazoles:  A New Class of Cytokine Suppressive Drugs with Low 5-Lipoxygenase and Cyclooxygenase Inhibitory Potency
Journal of Medicinal Chemistry·1996· 120 citedOpen Access
Use of Spin Echo Magic Angle Spinning <sup>1</sup>H NMR in Reaction Monitoring in Combinatorial Organic Synthesis
The Journal of Organic Chemistry·1996· 52 cited
2,4,5- triarylimidazole inhibitors of IL-1 biosynthesis
Bioorganic & Medicinal Chemistry Letters·1995· 132 cited
Resolution of hydroxyureas
Tetrahedron Letters·1993· 11 cited
ChemInform Abstract: An Efficient Conversion of Nitriles to Amidines.
ChemInform·1991
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Frequent Co-authors

Steven M. Weinreb(23), Jerry L. Adams(13), Margaret E. Sorenson(8), Don E. Griswold(5), John Breton(5), Jeffrey T. Laydon(4), John C. Lee(4), Jeffrey C. Boehm(4), Juanita M. Smietana(4), Timothy F. Gallagher(4), Marie Chabot‐Fletcher(4), David M. Tschaen(4), Masood Parvez(4), Peter L. Sheldrake(3), Susanta K. Sarkar(3), Edward F. Webb(3), George Seibel(2), Shouki Kassis(2), Dennis Lee(2), Susan M. Fier-Thompson(2)