Daniel Lesieur

Laboratoire de Chimie — France

Chemistry · Physical Sciences

31h-index2.8kcitations169works0.02yr avg
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Research Topics

Synthesis and Reactions of Organic Compounds(41), Circadian rhythm and melatonin(36), Synthesis and Biological Evaluation(36), Synthesis of heterocyclic compounds(27), Free Radicals and Antioxidants(21)

Publications169 total

Design and synthesis of 3-phenyltetrahydronaphthalenic derivatives as new selective MT2 melatoninergic ligands. Part II
Bioorganic & Medicinal Chemistry·2009· 27 cited
Synthesis of 3-phenylnaphthalenic derivatives as new selective MT2 melatoninergic ligands
Bioorganic & Medicinal Chemistry·2008· 26 citedOpen Access
Design and synthesis of benzofuranic derivatives as new ligands at the melatonin-binding site MT3
Bioorganic & Medicinal Chemistry·2008· 16 citedOpen Access
Homology modeling of MT1 and MT2 receptors
European Journal of Medicinal Chemistry·2008· 24 cited
Novel 1,3-dicarbonyl compounds having 2(3H)-benzazolonic heterocycles as PPARγ agonists
Bioorganic & Medicinal Chemistry·2006· 15 cited
Increased Susceptibility of Low-Density Lipoprotein to Ex Vivo Oxidation in Mice Transgenic for Human Apolipoprotein B Treated with 1 Melatonin-Related Compound Is Not Associated with Atherosclerosis Progression
Journal of Cardiovascular Pharmacology·2005· 14 cited
Pictet—Spengler Heterocyclizations via Microwave‐Assisted Degradation of DMSO.
ChemInform·2005· 2 cited
Pictet–Spengler heterocyclizations via microwave-assisted degradation of DMSO
Tetrahedron Letters·2005· 46 cited
Antioxidant activity of melatonin and a pinoline derivative on linoleate model system
Journal of Pineal Research·2005· 30 cited
Docking Study of Ligands into the Colchicine Binding Site of Tubulin
Journal of Enzyme Inhibition and Medicinal Chemistry·2004· 39 cited
Synthesis and Evaluation of Benzoxazolinonic Imidazoles and Derivatives as Non-steroidal Aromatase Inhibitors
Journal of Enzyme Inhibition and Medicinal Chemistry·2004· 14 citedOpen Access
New substrate analogues of human serotonin <i>N</i>‐acetyltransferase produce <i>in situ</i> specific and potent inhibitors
European Journal of Biochemistry·2003· 17 citedOpen Access
Molecular pharmacology of the ovine melatonin receptor: comparison with recombinant human MT1 and MT2 receptors
Biochemical Pharmacology·2003· 39 cited
New selective ligands of human cloned melatonin MT1 and MT2 receptors
Naunyn-Schmiedeberg s Archives of Pharmacology·2003· 243 cited
Protection of endogenous β-carotene in LDL oxidized by oxygen free radicals in the presence of supraphysiological concentrations of melatonin
Redox Report·2003· 10 citedOpen Access
Design, Synthesis and <i>In Vitro</i> Evaluation of Novel Benzo[<i>b</i>]thiophene Derivatives as Serotonin <i>N</i>-acetyltransferase (AANAT) Inhibitors
Journal of Enzyme Inhibition and Medicinal Chemistry·2003· 10 citedOpen Access
Therapeutic Perspectives for Melatonin Agonists and Antagonists
Journal of Neuroendocrinology·2003· 65 cited
Design and Synthesis of Naphthalenic Dimers as Selective MT<sub>1</sub>Melatoninergic Ligands
Journal of Medicinal Chemistry·2003· 61 citedOpen Access
Design and synthesis of 3-phenyl tetrahydronaphthalenic derivatives as new selective MT2 melatoninergic ligands
Bioorganic & Medicinal Chemistry·2003· 34 cited
Synthesis of 4-[4-(N,N-Dimethylsulfamoyl)piperazin-1-yl]quinolines Derivatives as Sorbitol Dehydrogenase Potential Inhibitors
Heterocycles·2003· 6 citedOpen Access
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Frequent Co-authors

Pierre Renard(17), Saı̈d Yous(16), Philippe Delagrange(14), Jean A. Boutin(13), Philippe Chavatte(8), Valérie Audinot(7), Caroline Bennejean(7), Béatrice Guardiola‐Lemaître(6), H.E. Howell(5), Pierre‐Yves Renard(5), Patrick Depreux(5), Patrick Duriez(5), Elisabeth Teissier(5), Pascal Berthelot(5), Anne Bonnaud(4), Peter J. Morgan(4), Bruno Pfeiffer(4), Daniel‐Henri Caignard(4), Andrea Gozzo(4), Jacques H. Poupaert(4)