Eliezer Falb

Chemistry · Physical Sciences

9h-index484citations20works0.02yr avg
OpenAlex↗ORCID↗Google Scholar↗

Accepting Students?

No reports yet. Know if this professor is taking students?

Research Topics

Carbohydrate Chemistry and Synthesis(4), Chemical Synthesis and Analysis(4), Synthesis and Biological Evaluation(4), Synthesis and Reactions of Organic Compounds(4), Asymmetric Synthesis and Catalysis(2)

Publications20 total

Introducing a Methyl Group into Pyridines and Quinolines: A Mini-Review
Heterocycles·2019· 1 citedOpen Access
An unusual rearrangement involving 5-bromo-1-phenylpyridone during its methyl cross coupling with turbo-Grignard reagent, leading to a 5-bromopyridone-fused seven-membered carbocyclic ring
Chemistry of Heterocyclic Compounds·2017· 1 cited
A highly efficient Suzuki–Miyaura methylation of pyridines leading to the drug pirfenidone and its CD<sub>3</sub> version (SD-560)
Green Chemistry·2017· 42 cited
Novel 5-Dimethylamino-1- and 2-Indanyl Uracil Derivatives
The Journal of Organic Chemistry·2006· 9 cited
In situ generation of Fmoc amino acid chlorides for extremely difficult couplings to sterically hindered secondary amines in solid-phase peptide synthesis
Kluwer Academic Publishers eBooks·2006
Cinnamic Acid Derived Oxazolinium Ions as Novel Cytotoxic Agents.
ChemInform·2002· 2 cited
Cinnamic acid derived oxazolinium ions as novel cytotoxic agents
European Journal of Medicinal Chemistry·2002· 18 cited
A bicyclic and hsst2 selective somatostatin analogue: design, synthesis, conformational analysis and binding
Bioorganic & Medicinal Chemistry·2001· 25 cited
ChemInform Abstract: From Amino Acids to Fused Chiral Pyrrolidines and Piperidines via the INOC Route.
ChemInform·2000
From Amino Acids to Fused Chiral Pyrrolidines and Piperidines via the INOC Route
European Journal of Organic Chemistry·2000· 15 cited
<i>In situ</i> generation of Fmoc‐amino acid chlorides using <i>bis</i>‐(trichloromethyl)carbonate and its utilization for difficult couplings in solid‐phase peptide synthesis
Journal of Peptide Research·1999· 145 cited
IOOC Route to Substituted Chiral Pyrrolidines. Potential Glycosidase Inhibitors
The Journal of Organic Chemistry·1998· 38 cited
ChemInform Abstract: Acetyl Chloride—Methanol as a Convenient Reagent for: A) Quantitative Formation of Amine Hydrochlorides, B) Carboxylate Ester Formation, C) Mild Removal of N‐Boc‐Protective Group.
ChemInform·1998· 1 cited
Acetyl Chloride-Methanol as a Convenient Reagent for: A) Quantitative Formation of Amine Hydrochlorides B) Carboxylate Ester Formation C) Mild Removal of N-t-Boc-Protective Group.
Synthetic Communications·1998· 107 cited
ChemInform Abstract: Hypoxic Radiosensitizers: Substituted Styryl Derivatives.
ChemInform·1995
ChemInform Abstract: Cycloadditions. Part 52. Utilization of L‐Serine in an Oxime Olefin Cycloaddition Route to a Functionalized Asymmetric Pyrrolidine, a Selective α‐Glucosidase Inhibitor.
ChemInform·1994
ChemInform Abstract: A Convenient Synthesis of Chiral Oxazolidin‐2‐ones and Thiazolidin‐2‐ ones and an Improved Preparation of Triphosgene.
ChemInform·1994
Utilization of L-serine in an oxime olefin cycloaddition route to a functionalized asymmetric pyrrolidine, a selective α-glucosidase inhibitor
Tetrahedron Letters·1994· 34 cited
Hypoxic Radiosensitizers: Substituted Styryl Derivatives
Archiv der Pharmazie·1994· 5 cited
A Convenient Synthesis of Chiral Oxazolidin-2-Ones and Thiazolidin-2-Ones and an Improved Preparation of Triphosgene
Synthetic Communications·1993· 41 cited

Frequent Co-authors

Abraham Nudelman(13), Alfred Häßner(10), Hugo E. Gottlieb(7), Tamar Yechezkel(3), Yosi Bechor(3), Konstantin Ulanenko(3), Amnon Albeck(3), Yoseph Salitra(2), Ayelet Nudelman(2), B. A. WEXLER(2), Andrey Tor(2), Michal Afri(2), Lilach Hedvati(2), B. O. Kraiz(2), R. A. Zhuk(2), Milon Sprecher(2), Yael Odesa(2), Naomi Shmueli‐Broide(2), C. Gi on(1), Bilha Fischer(1)