Adriaan P. IJzerman

Leiden University — Netherlands

Biochemistry, Genetics and Molecular Biology · Life Sciences

77h-index27.8kcitations635works2.12yr avg
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Research Topics

Receptor Mechanisms and Signaling(304), Adenosine and Purinergic Signaling(276), Pharmacological Receptor Mechanisms and Effects(110), Neuropeptides and Animal Physiology(108), Synthesis and Biological Evaluation(88)

Publications633 total

Adenosine receptors in GtoPdb v.2025.4
IUPHAR/BPS Guide to Pharmacology CITE·2025Open Access
Gonadotrophin-releasing hormone receptors in GtoPdb v.2025.3
IUPHAR/BPS Guide to Pharmacology CITE·2025Open Access
Hydroxycarboxylic acid receptors in GtoPdb v.2025.3
IUPHAR/BPS Guide to Pharmacology CITE·2025Open Access
Navigating Solute Carrier Transporters—A Comprehensive Review of Functionalized Small Molecule Probes for Target Identification and Characterization
Medicinal Research Reviews·2025Open Access
The solute carrier superfamily interactome
Molecular Systems Biology·2025· 9 citedOpen Access
Covalent functionalization of G protein-coupled receptors by small molecular probes
RSC Chemical Biology·2025Open Access
A patient-centric knowledge graph approach to prioritize mutants for selective anti-cancer targeting
2024Open Access
The solute carrier superfamily interactome
2024· 5 citedOpen Access
Author response for "Stereochemical optimization of <i>N</i>,2-substituted cycloalkylamines as norepinephrine reuptake inhibitors"
2024
Labeling of CC Chemokine Receptor 2 with a Versatile Intracellular Allosteric Probe
ACS Chemical Biology·2024· 1 citedOpen Access
Author response for "Stereochemical optimization of <i>N</i>,2-substituted cycloalkylamines as norepinephrine reuptake inhibitors"
2024
CC chemokine receptor 2 is allosterically modulated by sodium ions and amiloride derivatives through a distinct sodium ion binding site
Biochemical Pharmacology·2024
Advancing drug discovery through assay development: a survey of tool compounds within the human solute carrier superfamily
Frontiers in Pharmacology·2024· 9 citedOpen Access
<i>N</i>-Acyl-<i>N</i>-Alkyl Sulfonamide Probes for Ligand-Directed Covalent Labeling of GPCRs: The Adenosine A<sub>2B</sub> Receptor as Case Study
ACS Chemical Biology·2024· 7 citedOpen Access
Excuse me, there is a mutant in my bioactivity soup!A comprehensive analysis of the genetic variability landscape of bioactivity databases and its effect on activity modelling
2024· 3 citedOpen Access
Exploring novel dilazep derivatives as hENT1 inhibitors and potentially covalent molecular tools
Purinergic Signalling·2024· 3 citedOpen Access
Label-free detection of prostaglandin transporter (SLCO2A1) function and inhibition: insights by wound healing and TRACT assays
Frontiers in Pharmacology·2024· 4 citedOpen Access
Pharmacological characterization of allosteric modulators: A case for chemokine receptors
Medicinal Research Reviews·2024· 2 citedOpen Access
Accompanying data - Papyrus - A large scale curated dataset aimed at bioactivity predictions
Zenodo (CERN European Organization for Nuclear Research)·2024Open Access
Computational Characterization of Membrane Proteins as Anticancer Targets: Current Challenges and Opportunities
International Journal of Molecular Sciences·2024· 3 citedOpen Access
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Frequent Co-authors

Gerard J. P. van Westen(11), Laura H. Heitman(9), Margot W. Beukers(7), Kenneth A. Jacobson(6), Raymond C. Stevens(6), Herman van Vlijmen(6), Thea Mulder‐Krieger(6), Johannes Brussee(5), Vadim Cherezov(4), Vsevolod Katritch(4), Henk de Vries(4), Eelke B. Lenselink(4), Dong Guo(4), Andreas Bender(4), Jacobien K. von Frijtag Drabbe Künzel(4), Gye Won Han(3), S P H Alexander(3), Eamonn Kelly(3), Alistair Mathie(3), John A. Peters(3)