Michael P. Winters

Springhouse — United States

Pharmacology, Toxicology and Pharmaceutics · Life Sciences

17h-index2.8kcitations38works0.02yr avg
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Research Topics

Bioactive Compounds and Antitumor Agents(7), Chemical Synthesis and Analysis(5), Receptor Mechanisms and Signaling(5), Organic Chemistry Cycloaddition Reactions(5), Pain Mechanisms and Treatments(4)

Publications38 total

Discovery of a GPR40 Superagonist: The Impact of Aryl Propionic Acid α-Fluorination
ACS Medicinal Chemistry Letters·2018· 24 citedOpen Access
Discovery and optimization of a novel series of pyrazolyltetrahydropyran N-type calcium channel (Cav 2.2) blockers for the treatment of pain
Bioorganic & Medicinal Chemistry Letters·2018· 6 citedOpen Access
FFAR1 Agonism Restores Insulin Secretion in Rodents, Human Islets, and Diabetic Monkeys
Diabetes·2018· 1 cited
Therapeutic Potential of EP3 Receptor Antagonists for Treatment of Noninsulin Dependent Diabetes Mellitus across Multiple Preclinical Models
Diabetes·2018· 2 cited
Erratum to “Discovery of N-arylpyrroles as agonists of GPR120 for the treatment of type II diabetes” Bioorg. Med. Chem. Lett. 28 (2018) [841–846]
Bioorganic & Medicinal Chemistry Letters·2018· 1 cited
Discovery of N-arylpyrroles as agonists of GPR120 for the treatment of type II diabetes
Bioorganic & Medicinal Chemistry Letters·2018· 20 citedOpen Access
Discovery of novel benzo[b]thiophene tetrazoles as non-carboxylate GPR40 agonists
Bioorganic & Medicinal Chemistry Letters·2017· 15 cited
Design, synthesis and SAR of a novel series of heterocyclic phenylpropanoic acids as GPR120 agonists
Bioorganic & Medicinal Chemistry Letters·2017· 21 citedOpen Access
CCDC 931421: Experimental Crystal Structure Determination
The Cambridge Structural Database·2015Open Access
Lab-Scale Preparation of a Novel Cyclopenta[b]furan Chemokine Receptor Antagonist
Organic Process Research & Development·2014· 10 cited
ChemInform Abstract: Synthesis of Substituted 2,4,5,6‐Tetrahydrocyclopenta[c]pyrazoles and 2,4,5,6‐Tetrahydropyrrolo[3,4‐c]pyrazoles by Intramolecular Nitrilimine Cycloaddition.
ChemInform·2014
Discovery and SAR of a novel series of 2,4,5,6-tetrahydrocyclopenta[c]pyrazoles as N-type calcium channel inhibitors
Bioorganic & Medicinal Chemistry Letters·2014· 6 cited
Discovery and SAR of novel tetrahydropyrrolo[3,4-c]pyrazoles as inhibitors of the N-type calcium channel
Bioorganic & Medicinal Chemistry Letters·2014· 14 cited
The discovery and SAR of cyclopenta[b]furans as inhibitors of CCR2
Bioorganic & Medicinal Chemistry Letters·2014· 6 citedOpen Access
Synthesis of substituted 2,4,5,6-tetrahydrocyclopenta[c]pyrazoles and 2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazoles by intramolecular nitrilimine cycloaddition
Tetrahedron Letters·2014· 17 cited
A novel series of pyrazolylpiperidine N-type calcium channel blockers
Bioorganic & Medicinal Chemistry Letters·2012· 20 cited
Corrigendum to “Discovery, SAR and X-ray structure of 1H-benzimidazole-5-carboxylic acid cyclohexyl-methyl-amides as inhibitors of inducible T-cell kinase (Itk)” [Bioorg. Med. Chem. Lett. 18 (2008) 5545–5549]
Bioorganic & Medicinal Chemistry Letters·2009· 3 cited
5-Aminomethyl-1H-benzimidazoles as orally active inhibitors of inducible T-cell kinase (Itk)
Bioorganic & Medicinal Chemistry Letters·2008· 24 citedOpen Access
Discovery, SAR and X-ray structure of 1H-benzimidazole-5-carboxylic acid cyclohexyl-methyl-amides as inhibitors of inducible T-cell kinase (Itk)
Bioorganic & Medicinal Chemistry Letters·2008· 32 citedOpen Access
Itk kinase inhibitors: Initial efforts to improve the metabolical stability and the cell activity of the benzimidazole lead
Bioorganic & Medicinal Chemistry Letters·2008· 26 citedOpen Access
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Frequent Co-authors

Zhihua Sui(12), Harold W. Moore(7), Mark J. Wall(7), Mohammed A. Kashem(6), Hnin Hnin Khine(5), Steven S. Pullen(5), Gregory P. Roth(5), Mark R. Player(5), Nalin L. Subasinghe(5), Christopher A. Teleha(5), Dominic M. T. Chan(4), John P. Wolak(4), Ronald L. Magolda(4), Renée L. DesJarlais(4), Declan Ryan(4), Shuyuan Zhao(4), K.J.M. Moriarty(4), Hidenori Takahashi(4), Darius Robinson(4), James C. Lanter(4)