Andrzej J. Bojarski

Maj Institute of Pharmacology — Poland

Biochemistry, Genetics and Molecular Biology · Life Sciences

39h-index7.6kcitations381works2.72yr avg
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Research Topics

Receptor Mechanisms and Signaling(126), Synthesis and Biological Evaluation(74), Neurotransmitter Receptor Influence on Behavior(60), Computational Drug Discovery Methods(60), Neuroscience and Neuropharmacology Research(47)

Publications379 total

Chronic 5-HT7R activation drives depressive phenotypes and synaptic dysfunction
Acta Pharmacologica Sinica·2026
Fine-tuning 5-HT7 receptor selectivity, inverse agonism, and metabolic stability of new (aryloxy)ethyl-piperidines toward antidepressant and pro-cognitive properties
European Journal of Medicinal Chemistry·2025Open Access
The impact of secondary site interactions on the binding specificity of bitopic dopamine D2/D3 receptor ligands
European Journal of Medicinal Chemistry Reports·2025Open Access
Novel Dual 5-HT7 Antagonists and Sodium Channel Inhibitors as Potential Therapeutic Agents with Antidepressant and Anxiolytic Activities
Pharmaceuticals·2025Open Access
Intepirdine Derivatives Possessing Dual 5HT6 Antagonism / HDAC6 Inhibitory Activity
Chemistry - A European Journal·2025Open Access
Correction: Compound PZ-1262, a 4-isoquinoline-sulfonamide analog of Brexpiprazole, produces potential antidepressant, anxiolytic and procognitive effects in rodent models
Pharmacological Reports·2025Open Access
Identification of Orthosteric GABA<sub>B</sub> Receptor Ligands by Virtual Screening and <i>In Vitro</i> Validation
ACS Omega·2025Open Access
Compound PZ-1262, a 4-isoquinoline-sulfonamide analog of Brexpiprazole, produces potential antidepressant, anxiolytic and procognitive effects in rodent models
Pharmacological Reports·2025Open Access
Simultaneous 5-HT1BR agonist/5-HT6R antagonist action as a potential treatment of Parkinson’s disease and its comorbidities
Journal of Pharmacology and Experimental Therapeutics·2024· 5 citedOpen Access
Contilistat, a New Multitarget Small Polyfunctionalized Indole Derivative
Synlett·2024· 2 citedOpen Access
Design and Synthesis of Potential Multi-Target Antidepressants: Exploration of 1-(4-(7-Azaindole)-3,6-dihydropyridin-1-yl)alkyl-3-(1H-indol-3-yl)pyrrolidine-2,5-dione Derivatives with Affinity for the Serotonin Transporter
International Journal of Molecular Sciences·2024· 3 citedOpen Access
Contilisant+Tubastatin A Hybrids: Polyfunctionalized Indole Derivatives as New HDAC Inhibitor-Based Multitarget Small Molecules with <i>In Vitro</i> and <i>In Vivo</i> Activity in Neurodegenerative Diseases
Journal of Medicinal Chemistry·2024· 18 citedOpen Access
Unlocking the potential of higher-molecular-weight 5-HT7R ligands: Synthesis, affinity, and ADMET examination
Bioorganic Chemistry·2024· 4 citedOpen Access
Correction to: Unraveling psilocybin’s therapeutic potential: behavioral and neuroplasticity insights in Wistar-Kyoto and Wistar male rat models of treatment-resistant depression
Psychopharmacology·2024· 1 citedOpen Access
Uncovering the unique characteristics of different groups of 5-HT5AR ligands with reference to their interaction with the target protein
Pharmacological Reports·2024· 1 citedOpen Access
Unraveling psilocybin’s therapeutic potential: behavioral and neuroplasticity insights in Wistar-Kyoto and Wistar male rat models of treatment-resistant depression
Psychopharmacology·2024· 11 citedOpen Access
5-HT6 receptor neutral antagonists protect astrocytes: A lesson from 2-phenylpyrrole derivatives
European Journal of Medicinal Chemistry·2024· 2 citedOpen Access
Physicochemical, structural and biological characterisation of poly(3-hydroxyoctanoate) supplemented with diclofenac acid conjugates — Harnessing the potential in the construction of materials for skin regeneration processes
International Journal of Biological Macromolecules·2024· 7 citedOpen Access
5-Ht6 Receptor Neutral Antagonists Protect Astrocytes a Lesson from 2-Phenylpyrrole Derivatives
SSRN Electronic Journal·2024Open Access
Exploring the molecular basis of treatment-resistant depression: Discoveries from a rat model and psilocybin therapy
Neuroscience Applied·2024Open Access
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Frequent Co-authors

Grzegorz Satała(20), Paweł Zajdel(12), Anna Wesołowska(11), Anna Partyka(10), Maciej Pawłowski(9), Rafał Kurczab(9), Stefan Mordalski(7), Magdalena Jastrzębska‐Więsek(7), Krzysztof Marciniec(6), Krzysztof Rataj(5), Beata Duszyńska(5), Tomasz Lenda(5), Agata Siwek(5), Piotr Popik(5), Vittorio Canale(5), Christian Munk(4), Kasper Harpsøe(4), Alexander S. Hauser(4), David E. Gloriam(4), Marcin Kołaczkowski(4)